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BIBR 1532
BIBR 1532

Artikelnummer: Cay16608-10

BIBR 1532 is a mixed-type non-competitive inhibitor of telomerase (IC50 = 93 nM) that has little effect on several mammalian DNA and RNA polymerases, bacterial DNA helicase, or HIV-1 reverse transcriptase. It specifically targets the telomerase reverse transcriptase catalytic subunit, TERT. Through its effects on...
Schlagworte: Telomerase Inhibitor X, 2-[[(2E)-3-(2-naphthalenyl)-1-oxo-2-buten-1-yl]amino]-benzoic acid
Anwendung: Telomerase / TERT inhibitor
CAS 321674-73-1
MW: 331.4 D
ab 51,00 €
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NEU
BIBR 1532
BIBR 1532

Artikelnummer: TGM-T2380-100mg

Description: BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay). Target: Apoptosis, Telomerase. Smiles: C\C(=C/C(=O)Nc1ccccc1C(O)=O)c1ccc2ccccc2c1. References: Pascolo E, et al. J Biol Chem. 2002, 277(18), 15566-15572.
CAS 321674-73-1
MW: 331.36 D
ab 43,00 €
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