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LDN-27219
Artikelnummer: TGM-T11831-100mg
Description: LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM. Target: Others. Smiles: NNC(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1-c1ccccc1. References: Case A, et al. Kinetic analysis of the interaction of tissue transglutaminase with a nonpeptidic slow-binding inhibitor. Biochemistry. 2007 Jan 30,46(4):1106-15.
| Anwendung: | Tansglutaminase 2 (TG2) inhibitor |
| CAS | 312946-37-5 |
| MW: | 408.5 D |
ab 34,00 €
LDN-27219
Artikelnummer: Cay32975-1
LDN-27219 is an inhibitor of tissue transglutaminase 2 (TG2, IC50 = 0.25 µM) that promotes its closed conformation. LDN-27219 induces relaxation of isolated rat mesenteric arteries precontracted with the thromboxane receptor agonist U-46619 (Cay-16450) in a concentration-dependent manner, an effect that can be...
| Schlagworte: | 2-[(3,4-dihydro-4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)thio]-acetic acid, hydrazide (ACl) |
| Anwendung: | Tansglutaminase 2 (TG2) inhibitor |
| CAS | 312946-37-5 |
| MW: | 408.5 D |
ab 44,00 €
