Zu "288628-05-7" wurden 2 Artikel gefunden!
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STX-64
Artikelnummer: Cay9003206-1
STX-64 is a steroid sulfatase inhibitor (IC50 = 0.008 µM in placental microsomes). It also inhibits carbonic anhydrase II (CAII, IC50 = 0.025 µM). STX-64 inhibits LPS-induced production of nitric oxide (NO) and prostaglandin E2 (PGE2, Cay-14010) in RAW 264.7 macrophages (IC50s = 85.76 and 0.081 µM, respectively). It...
| Schlagworte: | 667 Coumate, BN83495, Irosustat, sulfamic acid, 6,7,8,9,10,11-hexahydro-6-oxobenzo[b]cyclohepta[d]pyran-3-yl ester |
| Anwendung: | Steroid sulfatase inhibitor |
| CAS | 288628-05-7 |
| MW: | 309.3 D |
ab 89,00 €
Irosustat
Artikelnummer: TGM-T4464-100mg
Description: Irosustat (667-Coumate) is a potent steroid sulfatase inhibitor, with an IC50 of 8 nM, and exhibits anti-breast cancer activity. Target: Others. Smiles: NS(=O)(=O)Oc1ccc2c3CCCCCc3c(=O)oc2c1. References: Raobaikady B,etal.Inhibition of MCF-7 breast cancer cell proliferation and in vivo steroid sulphatase...
| Schlagworte: | STX64 , BN83495 , 667-Coumate |
| Anwendung: | Targets steryl-sulfatase [EC:3.1.6.2] (STS) |
| CAS | 288628-05-7 |
| MW: | 309.34 D |
ab 30,00 €
