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KAT8 Inhibitor 19
KAT8 Inhibitor 19

Artikelnummer: Cay38977-5

KAT8 inhibitor 19 is an inhibitor of lysine acetyltransferase 8 (KAT8, IC50 = 12.1 µM). It is selective for KAT8 over KAT2A, KAT2B, KAT3B, KAT6A, and KAT7 at 200 µM. KAT8 (50 µM) reduces histone 4 lysine 16 acetylation (H4K16Ac) in HT-29 colorectal carcinoma cells. It reduces the viability of HCT116, H1299, A549,...
Schlagworte: Lysine Acetyltransferase 8 Inhibitor 19,...
Anwendung: KAT8 inhibitor
CAS 28532-21-0
MW: 295.3 D
ab 38,00 €
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MC4033
MC4033

Artikelnummer: TGM-T78156-100mg

Description: MC4033 is a selective lysine acetyltransferase 8 (KAT8) inhibitor (IC50: 12.1 µM) with anticancer effects, induces apoptosis, and can be used for the study of non-small cell lung cancer. Target: Histone Acetyltransferase, Apoptosis. Smiles: O=C(O)C1=CC=C(C=C1)N2N=C(C(=CC3=CC=CN3)C2=O)C. References:...
Anwendung: KAT8 inhibitor
CAS 28532-21-0
MW: 295.29 D
ab 30,00 €
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