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Torcetrapib
Torcetrapib

Artikelnummer: Cay15028-50

Torcetrapib is an inhibitor of cholesteryl ester transfer protein (CETP, IC50s = 47 and 51 nM for cholesteryl and triglyceride transfer, respectively). It is selective for CETP over phospholipid transfer protein (PLTP), lecithin:cholesterol acyltransferase (LCAT), and hepatic and lipoprotein lipases at 10 µM....
Schlagworte: CP 529,414,...
Anwendung: CETP inhibitor
CAS 262352-17-0
MW: 600.5 D
ab 149,00 €
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NEU
Torcetrapib
Torcetrapib

Artikelnummer: TGM-T2499-10mg

Description: Torcetrapib (CP-529414) is a cholesteryl ester transfer protein (CETP) inhibitor designed to reduce the heterotypic transfer of cholesteryl ester from HDL to LDL and/or VLDL. It failed in phase III trials due to an excess of deaths. Target: CETP. Smiles:...
Schlagworte: CP-529414
Anwendung: Targets cholesteryl ester transfer protein (CETP)
CAS 262352-17-0
MW: 600.47 D
ab 30,00 €
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