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alphavbeta5 Integrin-IN-1
alphavbeta5 Integrin-IN-1

Artikelnummer: Cay39733-1

alphavbeta5 Integrin-IN-1 is an inhibitor of alphaVbeta5 integrin (IC50 = 0.0063 µM). It is selective for alphaVbeta5 over alphaVbeta1, alphaVbeta3, alphaVbeta6, and alphaVbeta8 (IC50s = 2.51, 5.01, 50.1, and 50.1 µM, respectively). alphavbeta5 Integrin-IN-1 inhibits adhesion of alphaVbeta5-expressing K562 cells to...
Schlagworte: alphavbeta5 Integrin Inhibitor 1,...
Anwendung: AlphaVbeta5 integrin inhibitor
CAS 2615912-33-7
MW: 475.5 D
441,00 €
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alphavbeta5 integrin-IN-1
alphavbeta5 integrin-IN-1

Artikelnummer: TGM-T40243-1mg

Description: alphavbeta5 integrin-IN-1, a potent and selective alphavbeta5 integrin inhibitor, exhibits a high inhibitory potency with a pIC50 value of 8.2. Target: Others. Smiles: OC(=O)C[C@H](C(=O)N1CC[C@@H](CCC2=CC=C3CCCN=C3N2)C1)c1cccc(c1)C(F)(F)F , c:20,t:13,15, . References: Lippa RA, et al. Discovery of the...
Anwendung: AlphaVbeta5 integrin inhibitor
CAS 2615912-33-7
MW: 475.512 D
1.013,00 €
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