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Anamorelin
Anamorelin

Artikelnummer: TGM-T10319-10mg

Description: Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). Target: GHSR. Smiles: CN(C)N(C)C(=O)[C@@]1(Cc2ccccc2)CCCN(C1)C(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)(C)N. References: Pietra C, et al. Anamorelin HCl (ONO-7643), a novel ghrelin receptor agonist, for the...
Schlagworte: ONO-7643, RC-1291
CAS 249921-19-5
MW: 546.7 D
ab 55,00 €
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Anamorelin
Anamorelin

Artikelnummer: Cay24676-10

Anamorelin is a small molecule agonist of the growth hormone (GH) secretagogue receptor 1a (GHS-R1a) and a mimetic of ghrelin (Cay-15072, Cay-24458, Ki = 0.7 nM). It induces calcium mobilization in CHO cells expressing rat GHS-R1a in a concentration-dependent manner and GH release from rat pituitary cells (EC50 =...
Schlagworte: RC-1291,...
Anwendung: GHSR/ ghrelin receptor agonist
CAS 249921-19-5
MW: 546.7 D
ab 94,00 €
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