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SGC-GAK-1
Artikelnummer: Cay33229-5
SGC-GAK-1 is an inhibitor of cyclin G-associated kinase (GAK, Ki = 3.1 nM). It is greater than 50-fold selective for GAK over a panel of 400 kinases at 1 µM but does bind to RIPK2 in a bioluminescence resonance energy transfer (BRET) engagement assay (IC50 = 360 nM). SCG-GAK-1 reduces the viability of LNCaP and...
| Schlagworte: | 6-bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine |
| Anwendung: | GAK inhibitor |
| CAS | 2226517-76-4 |
| MW: | 389.2 D |
ab 58,00 €
SGC-GAK-1
Artikelnummer: TGM-T5169-100mg
Description: SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM). Target: Serine/threonin kinase. Smiles: COc1cc(Nc2ccnc3ccc(Br)cc23)cc(OC)c1OC. References: Asquith CRM, et al. SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK). J Med Chem. 2019 Feb 26.
| Anwendung: | GAK inhibitor |
| CAS | 2226517-76-4 |
| MW: | 389.24 D |
ab 41,00 €
