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ARV-110
ARV-110

Artikelnummer: Cay39662-25

ARV-110 is a proteolysis-targeting chimera (PROTAC) that contains a cereblon ligand 1-derivative connected to an androgen receptor (AR) ligand by a linker region. It reduces AR levels in VCaP prostate cancer cells in a time- and concentration-dependent manner. ARV-110 (1 µM) decreases VCaP cancer cell proliferation....
Schlagworte: Bavdegalutamide,...
Anwendung: PROTAC, AR degradation
CAS 2222112-77-6
MW: 812.3 D
ab 81,00 €
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Bavdegalutamide
Bavdegalutamide

Artikelnummer: TGM-T22263-100mg

Description: Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR). Bavdegalutamide can be used in studies about prostate cancer. Bavdegalutamide shows oral activity and selectivity and facilitates the ubiquitination and degradation of AR. Target: Androgen Receptor. Smiles:...
Schlagworte: ARV-110
Anwendung: Targets androgen receptor (AR, NR3C4)
CAS 2222112-77-6
MW: 812.29 D
ab 84,00 €
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ARV-110
ARV-110

Artikelnummer: BPS-82037

ARV-110 is an androgen receptor PROTAC degrader. It promotes ubiquitination and degradation of the androgen receptor.
Anwendung: Protac(R) reagent
CAS 2222112-77-6
MW: 812,3 D
1.343,00 €
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