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PFI-653
PFI-653

Artikelnummer: Cay40955-10

PFI-653 is an inhibitor of the pantetheinase vanin-1 (IC50 = 6.85 nM for the human enzyme). In vivo, PFI-653 (50 mg/kg) prevents reductions in body weight, as well as reduces disease severity and serum vanin-1 levels in a mouse model of colitis induced by dextran sulfate sodium (DSS, Cay-23250). See the Structural...
Schlagworte: Vanin 1 Inhibitor 1, Vanin 1-IN-1, VNN1 Inhibitor 1, VNN1-IN-1,...
Anwendung: Vanin-1 inhibitor
CAS 2173134-00-2
MW: 354.4 D
ab 83,00 €
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Vanin-1-IN-1
Vanin-1-IN-1

Artikelnummer: TGM-T8218-100mg

Description: Vanin-1-IN-1 (VUN34002) is an vanin-1 enzyme inhibitor. Target: Others. Smiles: O=C(N1CCC2(C1)CCOCC2)c1cnc(NCc2cnccn2)nc1. References: Agustin Casimiro-Garcia, et al. Novel pyrimidine carboxamides as inhibitors of vanin-1 enzyme. WO2018011681A1.
Schlagworte: VUN34002
Anwendung: Vanin-1 inhibitor
CAS 2173134-00-2
MW: 354.41 D
ab 46,00 €
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