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MA-0204
MA-0204

Artikelnummer: TGM-T15945-100mg

Description: MA-0204 is a highly selective and orally available peroxisome proliferator-activated receptor delta (PPARdelta) modulator (EC50s: 0.4 nM, 7.9 nM and 10 nM for human, mouse and rat PPARdelta, respectively). It is a potential treatment for Duchene Muscular Dystrophy (DMD). Target: PPAR. Smiles:...
Anwendung: PPARdelta agonist
CAS 2095128-17-7
MW: 476.49 D
ab 88,00 €
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MA-0204
MA-0204

Artikelnummer: Cay26025-1

MA-0204 is an agonist of peroxisome proliferator-activated receptor delta (PPARdelta). It selectively induces reporter gene expression in CV-1 cells expressing human PPARdelta (EC50 = 0.4 nM) over CV-1 cells expressing human PPARalpha or PPARgamma (EC50s = 6,990 and >10,000 nM, respectively). MA-0204 increases the...
Schlagworte: 3R-methyl-6-[2-[[5-methyl-2-[4-(trifluoromethoxy)phenyl]-1H-imidazol-1-yl]methyl]phenoxy]-hexanoic acid
Anwendung: PPARdelta agonist
CAS 2095128-17-7
MW: 476.5 D
ab 239,00 €
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