Zu "209268-36-0" wurden 2 Artikel gefunden!
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S-5751
Artikelnummer: TGM-T28651-1mg
Description: S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma. Target: Others. Smiles: N(C(=O)C=1C=2C(SC1)=CC=C(O)C2)[C@H]3[C@]4(C(C)(C)[C@](C4)(C[C@@H]3C/C=C\CCCC(O)=O)[H])[H]. References: Arimura A, Yasui K, Kishino J, Asanuma F, Hasegawa H, Kakudo S, Ohtani M,...
| Schlagworte: | S 5751 |
| Anwendung: | Prostaglandin D2 receptor (PTGDR) antagonist |
| CAS | 209268-36-0 |
| MW: | 441.58 D |
ab 122,00 €
S-5751
Artikelnummer: Cay10004030-5
S-5751 is an antagonist of the prostaglandin D2 (PGD2) receptor DP1 (Ki = 1.6 nM) that shows at least 20-fold selectivity over receptors for thromboxane and prostacyclin, as well as the PGE2 receptor EP2. Orally administered S-5751 blocks PGD2-induced plasma exudation in the conjunctiva (ED50 = 0.099 mg/kg) and...
| Schlagworte: | (5Z)-7-[(1R,2R,3S,5S)-2-[[(5-hydroxybenzo[b]thien-3-yl)carbonyl]amino]-6,6-dimethylbicyclo[3.1.1]hept-3-yl]-5-heptenoic acid |
| Anwendung: | Prostaglandin D2 receptor (PTGDR) antagonist |
| CAS | 209268-36-0 |
| MW: | 441.6 D |
ab 67,00 €
