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Casein Kinase Inhibitor A51
Casein Kinase Inhibitor A51

Artikelnummer: Cay44831-1

Casein kinase inhibitor A51 is an inhibitor of casein kinase 1alpha (CK1alpha). It binds to CK1alpha, CK1delta, and CK1epsilon (Kds = 5.3, 1.8, and 4.4 nM, respectively) and reduces phosphorylation of beta-catenin at serine 45, a site phosphorylated specifically by CK1alpha, when used at a concentration of 1 µM....
Schlagworte: BTX-A51, trans-N-[5-chloro-4-[5-(cyclopropylmethyl)-1-methyl-1H-pyrazol-4-yl]-2-pyrimidinyl]-1,4-cyclohexanediamine
Anwendung: CK1alpha inhibitor
CAS 2079068-74-7
MW: 360.89 D
ab 69,00 €
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Casein Kinase inhibitor A51
Casein Kinase inhibitor A51

Artikelnummer: TGM-T9175-2mg

Description: Casein Kinase inhibitor A51 is an orally active casein kinase 1alpha (CK1alpha) inhibitor with anticancer activity that induces apoptosis in leukemia cells, and may be used in the study of neck cancers, acute myeloid leukemia, breast and prostate cancers. Target: Casein Kinase, Apoptosis, CDK. Smiles:...
Anwendung: Casein Kinase inhibitor
CAS 2079068-74-7
MW: 360.88 D
ab 73,00 €
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