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NI-42
Artikelnummer: Cay28293-5
NI-42 is an inhibitor of the bromodomain and PHD finger-containing 1 (BRPF1) bromodomain (IC50 = 7.9 nM). It is selective for BRPF1 over BRPF2/BRD1, BRPF3, BRD9, and BRD4/BD1 (IC50s = 48, 260, 310, and 4,500 nM, respectively). NI-42 inhibits the growth of OCI-AML2, Nomo-1, THP-1, KG-1, and MV-4-11 acute myeloid...
| Schlagworte: | 4-cyano-N-(1,2-dihydro-1,3-dimethyl-2-oxo-6-quinolinyl)-benzenesulfonamide |
| Anwendung: | Peregrin/BRPF1 inhibitor |
| CAS | 1884640-99-6 |
| MW: | 353.4 D |
ab 51,00 €
NEU
NI-42
Artikelnummer: TGM-T16321-100mg
Description: NI-42 is a structurally orthogonal chemical probe for the BRPFs and is biased. It effective inhibitor of the BRD of the BRPFs (IC50s of BRPF1/2/3=7.9/48/260 nM, Kds of BRPF1/2/3=40/210/940 nM). It also has excellent selectivity over nonclass IV BRD proteins. Target: Epigenetic Reader Domain. Smiles:...
| Anwendung: | Peregrin/BRPF1 inhibitor |
| CAS | 1884640-99-6 |
| MW: | 353.39 D |
ab 37,00 €
