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(5Z,2E)-CU-3
Artikelnummer: TGM-T10177-100mg
Description: (5Z,2E)-CU-3 is a potent and highly selective inhibitor of the DGKalpha isozyme with an IC50 value of 0.6 µM, competing with ATP and exhibiting a Km value of 0.48 mM. It specifically targets the catalytic region of DGKalpha without affecting the regulatory region and has demonstrated antitumor and...
| CAS | 1815598-71-0 |
| MW: | 392.47 D |
ab 39,00 €
(5Z,2E)-CU-3
Artikelnummer: Cay37770-1
(5Z,2E)-CU-3 is an inhibitor of diacylglycerol kinase alpha (DGK-alpha, IC50 = 0.6 µM for the porcine enzyme). It is selective for DGK-alpha over other type I DGKs, as well as type II, type III, type IV, and type V DGKs (IC50s = 7-36 µM). (5Z,2E)-CU-3 (5 µM) induces apoptosis in HeLa cervical and HepG2 liver cancer...
| Schlagworte: | N-[(5Z)-5-[(2E)-3-(2-furanyl)-2-propen-1-ylidene]-4-oxo-2-thioxo-3-thiazolidinyl]-benzenesulfonamide |
| Anwendung: | DGK-alpha inhibitor |
| CAS | 1815598-71-0 |
| MW: | 392.5 D |
ab 44,00 €
