Zu "174635-53-1" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
SB-218795
Artikelnummer: Cay42373-10
An NK3 receptor antagonist (Ki = 0.013 µM), selective for NK3 over NK1 and NK2 receptors (Kis = >100 and 1.221 µM, respectively), inhibits senktide-induced contractions in isolated rabbit iris sphincter muscle preparations (Kb = 43 nM), inhibits substance P-induced contraction of longitudinal and circular smooth...
| Schlagworte: | aR-[[(2-phenyl-4-quinolinyl)carbonyl]amino]-benzeneacetic acid, methyl ester |
| Anwendung: | NK3 receptor (TACR3) antagonist |
| CAS | 174635-53-1 |
| MW: | 396.44 D |
ab 133,00 €
SB 218795
Artikelnummer: TGM-T23316-100mg
Description: SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1. Target: Neurokinin receptor. Smiles: C(N[C@@H](C(OC)=O)C1=CC=CC=C1)(=O)C=2C3=C(N=C(C2)C4=CC=CC=C4)C=CC=C3. References: Medhurst AD, et, al. In vitro and...
| CAS | 174635-53-1 |
| MW: | 396.44 D |
ab 42,00 €
