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JZP 361
Artikelnummer: Cay43994-10
JZP 361 is an inhibitor of monoacylglycerol lipase (MAGL, IC50 = 46 nM). It is selective for MAGL over fatty acid amide hydrolase (FAAH) and alpha/beta-hydrolase domain-containing protein 6 (ABHD6, IC50s = 7,240 and 1,790 nM, respectively). JZP 361 also antagonizes histamine activity in isolated guinea pig ileum...
| Schlagworte: | [4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl]-1H-1,2,4-triazol-1-yl-methanone |
| Anwendung: | Monoglyceride lipase inhibitor |
| CAS | 1680193-80-9 |
| MW: | 405.89 D |
ab 116,00 €
JZP-361
Artikelnummer: TGM-T27703-100mg
Description: JZP-361 is a specific MAGL inhibitor with IC50s of 46 nM, 7.24 µM, and 1.79 µM for human recombinant MAGL, human recombinant FAAH, and human hABHD6. JZP-361 displays anti-histaminergic activities. JZP-361 can be used in studies about asthma. Target: MAGL, Histamine Receptor, Lipase. Smiles:...
| Schlagworte: | JZP361 , JZP 361 |
| CAS | 1680193-80-9 |
| MW: | 405.88 D |
ab 37,00 €
