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Tavapadon
Tavapadon

Artikelnummer: TGM-T16999-100mg

Description: Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist. Target: Dopamine Receptor. Smiles: CC1=C(C=CC(OC2=C(C(F)(F)F)C=CC=N2)=C1)C3=C(C)C(=O)NC(=O)N3C. References: Young D, et al. D1 Agonist Improved Movement of Parkinsonian Nonhuman Primates with Limited...
Schlagworte: PF-6649751, CVL-751
Anwendung: Targets dopamine receptor D1 (DRD1)
CAS 1643489-24-0
MW: 391.34 D
ab 74,00 €
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PF-06649751
PF-06649751

Artikelnummer: Cay33556-10

PF-06649751 is a dopamine D1 and D5 receptor partial agonist. It increases locomotor activity and reduces a global parkinsonian disability score in a macaque model of Parkinson's disease induced by MPTP when administered at a dose of 0.04 mg/kg.Formal Name:...
Schlagworte: CVL-751, 1,5-dimethyl-6-[2-methyl-4-[[3-(trifluoromethyl)-2-pyridinyl]oxy]phenyl]-2,4(1H,3H)-pyrimidinedione
Anwendung: Dopamine D1 / D5 receptor partial agonist
CAS 1643489-24-0
MW: 391.3 D
ab 55,00 €
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