Zu "1621175-65-2" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
TC-G-1008
Artikelnummer: TGM-T4648-100mg
Description: TC-G-1008 (GPR39-C3) is a zinc receptor agonist with EC50 values of 0.4 nM for rat GPR39 and 0.8 nM for human GPR39. Target: GHSR. Smiles: CNc1nc(NCc2ccc(NS(C)(=O)=O)cc2Cl)cc(n1)-c1ccccn1. References: Peukert S, et al. Discovery of 2-Pyridylpyrimidines as the First Orally Bioavailable GPR39 Agonists....
| Schlagworte: | GPR39-C3 |
| Anwendung: | GPR39 agonist |
| CAS | 1621175-65-2 |
| MW: | 418.9 D |
ab 42,00 €
GPR39-C3
Artikelnummer: Cay25445-1
GPR39-C3 is a potent agonist of the orphan G protein-coupled receptor GPR39 with EC50 values of 0.8 and 0.4 nM for cAMP production in HEK293 cells expressing human and rat receptors, respectively. It is selective for GPR39 over a panel of kinases (IC50s = >10 µM), ghrelin and neurotensin-1 receptors (IC50s = >30...
| Schlagworte: | N-[3-chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]-methanesulfonamide |
| Anwendung: | GPR39 agonist |
| CAS | 1621175-65-2 |
| MW: | 418.9 D |
ab 45,00 €
