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L-371,257
Artikelnummer: Cay42436-1
A nonpeptide oxytocin receptor antagonist (Ki = 19 and 4.6 nM for the rat uterine and human uterine receptors, respectively), selective for oxytocin receptors over human AVP receptors V1A and -V2 (Kis = 3,200 and >10,000 nM for the human platelet and kidney receptors, respectively) and rat AVP receptor V2 (Ki =...
| Schlagworte: | 1-[1-[4-[(1-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]-4-piperidinyl]-1,4-dihydro-2H-3,1-benzoxazin-2-one |
| Anwendung: | Nonpeptide oxytocin receptor antagonist |
| CAS | 162042-44-6 |
| MW: | 507.6 D |
ab 40,00 €
L-371,257
Artikelnummer: TGM-T15682-100mg
Description: L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a. Target: Oxytocin Receptor, Vasopressin Receptor. Smiles: COc1cc(OC2CCN(CC2)C(C)=O)ccc1C(=O)N1CCC(CC1)N1C(=O)OCc2ccccc12. References: Williams PD, et...
| CAS | 162042-44-6 |
| MW: | 507.58 D |
ab 33,00 €
