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Thioperamide maleate
Artikelnummer: TGM-T41247-10mg
Description: Thioperamide maleate (MR-12842 maleate) is an effective and selective H3 receptor antagonist (Ki = 4.3 nM) that inhibits [3H]histamine synthesis (Ki = 31 nM). Target: Histamine Receptor. Smiles: OC(=O)\C=C/C(O)=O.S=C(NC1CCCCC1)N1CCC(CC1)c1cnc[nH]1. References: Na Wang, et al. Histamine H3 Receptor...
| Schlagworte: | MR-12842 maleate |
| Anwendung: | Histamine H3 receptor antagonist |
| CAS | 148440-81-7 |
| MW: | 408.52 D |
ab 37,00 €
Thioperamide (maleate)
Artikelnummer: Cay10011127-1
Thioperamide (maleate) is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier. This compound binds to rat cerebral cortical cells in vitro with a pKi value of 8.4 and inhibits histamine binding in vivo with an ED50 value of 1 mg/kg. At a dose of 5 mg/kg thioperamide (maleate) inhibits...
| Schlagworte: | N-cyclohexyl-4-(1H-imidazol-5-yl)-1-piperidinecarbothioamide, 2Z-butenedioate |
| Anwendung: | Histamine H3 receptor antagonist |
| CAS | 148440-81-7 |
| MW: | 408.5 D |
ab 21,00 €
