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MS436
MS436

Artikelnummer: LKT-M7200.1

BRD4 inhibitor.
Anwendung: BRD4 inhibitor
CAS 1395084-25-9
MW: 383.43 D
ab 128,00 €
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MS436
MS436

Artikelnummer: TGM-T1854-100mg

Description: MS436 is a selective, small-molecule inhibitor for the BRD4 bromodomains. Target: Epigenetic Reader Domain. Smiles: Cc1cc(\N=N\c2ccc(cc2)S(=O)(=O)Nc2ccccn2)c(N)cc1O. References: Zhang G, et al. J Med Chem. 2013, 56(22), 9251-9264.
Anwendung: Bromodomain inhibitor, BRD4 inhibitor
CAS 1395084-25-9
MW: 383.42 D
ab 36,00 €
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MS-436
MS-436

Artikelnummer: BPS-82061-1

MS-436, through a set of water-mediated interactions, exhibits low nanomolar affinity (estimated Ki of 30-50 nM) to BRD4 with preference for the first bromodomain over the second. MS-436 effectively blocks BRD4 transcriptional activity in lipopolysaccharide-induced production of both nitric oxide and IL-6 in mouse...
Schlagworte: MS436, MS 436,
Anwendung: Bromodomain inhibitor, BRD4 inhibitor
CAS 1395084-25-9
MW: 383,4 D
ab 1.228,00 €
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