Zu "1321924-70-2" wurden 3 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
VTX-27
Artikelnummer: SYN-1206-M001
Soluble in DMSO. VTX-27 is a potent and selective inhibitor of the PKCtheta enzyme, with over 1000-fold against classical isoforms and over 10000-fold against atypical isoforms. Target: PKC theta
| Schlagworte: | VTX27 |
| Anwendung: | PKC theta inhibitor |
| CAS | 1321924-70-2 |
| MW: | 418,9 D |
ab 339,00 €
VTX-27
Artikelnummer: TGM-T13314-100mg
Description: VTX-27 is a selective inhibitor of protein kinase C theta (PKC theta) (Kis: 0.08 nM and 16 nM for PKC theta and PKC delta). Target: PKC. Smiles: FC1=C(C=2C=3C(NN2)=NC=CC3)N=C(C(Cl)=C1)N4C[C@@]([C@](C(C)C)(C)O)(NCC4)[H]. References: Jimenez JM, et al. Design and optimization of selective protein kinase C...
| Anwendung: | PKCtheta inhibitor |
| CAS | 1321924-70-2 |
| MW: | 418.9 D |
ab 80,00 €
VTX-27
Artikelnummer: Cay36938-1
VTX-27 is a PKCtheta inhibitor (Ki = 0.08 nM). It is selective for PKCtheta over PKCalpha, -betaI, -betaII, -gamma, -delta, -epsilon, -eta, -µ, and -zeta with Ki values ranging from 1 to >5,000 nM as well as a panel of seven kinases from the Src, spleen tyrosine kinase (Syk), Tec, and MAP kinase families (Kis =...
| Schlagworte: | (alphaR,2S)-4-[3-chloro-5-fluoro-6-(1H-pyrazolo[3,4-b]pyridin-3-yl)-2-pyridinyl]-alpha-methyl-alpha-(1-methylethyl)-2-pipe... |
| Anwendung: | PKCtheta inhibitor |
| CAS | 1321924-70-2 |
| MW: | 418.9 D |
ab 143,00 €
