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CYM2503
Artikelnummer: TGM-T8963-100mg
Description: CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by its inability to displace iodinated galanin, or to induce IP1 accumulation on its...
| Anwendung: | GAL2 receptor positive allosteric modulator |
| CAS | 1308833-36-4 |
| MW: | 777.95 D |
ab 31,00 €
CYM 2503
Artikelnummer: Cay36590-1
CYM 2503 is a positive allosteric modulator (PAM) of the galanin-2 (GAL2) receptor. It enhances the production of inositol monophosphate (IP1) induced by galanin in HEK293 cells expressing the GAL2 receptor (EC50 = 0.69 µM). CYM 2503 (60 mg/kg) increases the latency to first electrographic and behavioral seizures...
| Schlagworte: | 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(1,2-dihydro-4-methyl-2-oxo-7-quinolinyl)-N6-[(1,1-dimethylet... |
| Anwendung: | GAL2 receptor positive allosteric modulator |
| CAS | 1308833-36-4 |
| MW: | 778 D |
ab 49,00 €
