Zu "1282512-48-4" wurden 4 Artikel gefunden!

Für die Filterung wurden keine Ergebnisse gefunden!
GDC-0032
GDC-0032

Artikelnummer: Cay17387-1

GDC-0032 is a potent inhibitor of phosphatidylinositol 3-kinase (PI3K) isoforms alpha, delta, and gamma (IC50s = 0.28, 0.12, and 0.97 nM, respectively) that is 31 times less potent at PI3Kbeta. It is over 1,000-fold selective for p100alpha over other PI3K-like kinases, including DNA-dependent protein kinase...
Schlagworte: Taselisib,...
Anwendung: PI3K alpha, delta, gamma inhibitor
CAS 1282512-48-4
MW: 460.5 D
ab 58,00 €
Bewerten
GDC-0032
GDC-0032

Artikelnummer: SYN-1202-M001

Slightly soluble ( 10 fold selective over PI3Kbeta Target: PI3K , Kinase Group: Lipid Kinases , Substrate: Lipid
Schlagworte: GDC0032
Anwendung: PI3K alpha / delta / gamma inhibitor
CAS 1282512-48-4
MW: 460,5 D
ab 123,00 €
Bewerten
GDC-0032
GDC-0032

Artikelnummer: LKT-G1308.1

PI3K inhibitor.
Schlagworte: GDC0032, Taselisib
Anwendung: PI3K alpha, delta, gamma inhibitor
CAS 1282512-48-4
MW: 460.53 D
ab 75,00 €
Bewerten
Taselisib
Taselisib

Artikelnummer: TGM-T1999-100mg

Description: Taselisib (GDC-0032) is an orally bioavailable inhibitor of the class I phosphatidylinositol 3-kinase (PI3K) alpha isoform (PIK3CA), with potential antineoplastic activity. Target: PI3K, Carbonic Anhydrase. Smiles: CC(C)n1nc(C)nc1-c1cn2CCOc3cc(ccc3-c2n1)-c1cnn(c1)C(C)(C)C(N)=O. References: Ndubaku CO,...
Schlagworte: GDC-0032, RG-7604
CAS 1282512-48-4
MW: 460.53 D
ab 37,00 €
Bewerten