Zu "1203490-23-6" wurden 2 Artikel gefunden!
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Ralaniten
Artikelnummer: Cay42391-10
An antagonist of the androgen receptor NTD, inhibits androgen receptor NTD transactivation in a reporter assay (IC50 = 7.4 µM), reduces androgen-dependent growth of LNCaP cells from 10-30 µM, decreases tumor volume in an LNCaP CRPC mouse xenograft model at 50 mg/kg. Formulation: A solid. InChI:...
| Schlagworte: | EPI-002, (2R)-3-[4-[1-[4-[(2S)-3-chloro-2-hydroxypropoxy]phenyl]-1-methylethyl]phenoxy]-1,2-propanediol |
| Anwendung: | Androgen receptor NTD antagonist |
| CAS | 1203490-23-6 |
| MW: | 394.89 D |
ab 142,00 €
Ralaniten
Artikelnummer: TGM-T28502-100mg
Description: Ralaniten (EPI-002) is a potent, specific, and orally active antagonist of the androgen receptor N-terminal structural domain (AR-NTD), inhibiting AR transcriptional activity with an IC50 value of 7.4 µM. Ralaniten exhibits anticancer activity and is used to study desmoplasia-resistant prostate cancer...
| Schlagworte: | EPI-002 |
| Anwendung: | Targets androgen receptor (AR, NR3C4) |
| CAS | 1203490-23-6 |
| MW: | 394.89 D |
ab 33,00 €
