Zu "1169755-45-6" wurden 2 Artikel gefunden!
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INDY
Artikelnummer: AG-CR1-3665-M005
White to off-white solid. Soluble in DMSO (10mg/ml). Potent and selective ATP-competitive DYRK1A and DYRK1B inhibitor (IC50=240nM and 230nM respectively). Binds at the ATP-binding cleft of the enzyme, Inhibits also DYRK2, DYRK3, CLK1, CLK4, casein kinase 1 (CSNK1D) and PIM1 (>90% inhibition at the same...
| Schlagworte: | (1Z)-1-(3-Ethyl-5-hydroxy-2(3H)-benzothiazolylidene)-2-propanone |
| Anwendung: | Potent selective ATP-competitive DYRK1A / DYRK1B inhibitor |
| CAS | 1169755-45-6 |
| MW: | 235,3 D |
88,00 €
INDY
Artikelnummer: Cay23895-1
INDY is an ATP-competitive inhibitor of dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A (DYRK1A, Ki = 180 nM, IC50 = 240 nM). It is selective for DYRK1A over monoamine oxidase (MAO) A and B at concentrations up to 100 µM. INDY inhibits DYRK1A phosphorylation of tau in COS-7 cells expressing...
| Schlagworte: | 1Z-(3-ethyl-5-hydroxy-2(3H)-benzothiazolylidene)-2-propanone |
| Anwendung: | DYRK1A inhibitor |
| CAS | 1169755-45-6 |
| MW: | 235.3 D |
ab 40,00 €
