Zu "1164462-05-8" wurden 2 Artikel gefunden!

Für die Filterung wurden keine Ergebnisse gefunden!
TG4-155
TG4-155

Artikelnummer: TGM-T5482-100mg

Description: TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less effective at EP4 (KB = 11.4 µM) and a panel of other receptors and channels. Target: Prostaglandin Receptor. Smiles: COc1cc(\C=C\C(=O)NCCn2c(C)cc3ccccc23)cc(OC)c1OC. References: Jiang J , Ganesh T , Du Y , et al. Small...
Anwendung: Brain penetrant EP2 antagonist
CAS 1164462-05-8
MW: 394.46 D
ab 31,00 €
Bewerten
TG4-155
TG4-155

Artikelnummer: Cay17639-10

Prostaglandin E2 (PGE2) evokes distinct responses through four different 'E prostanoid' (EP) receptors. EP2 is a G protein-coupled receptor that has diverse roles, including those in cancer, inflammation, and neuroprotection. TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less...
Schlagworte: (2E)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide
Anwendung: Brain penetrant EP2 antagonist
CAS 1164462-05-8
MW: 394.5 D
ab 85,00 €
Bewerten