Zu "1054-88-2" wurden 2 Artikel gefunden!
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Spiroxatrine
Artikelnummer: Cay33415-10
Spiroxatrine is an antagonist of the serotonin (5-HT) receptor subtype 5-HT1A (Ki = 3 nM) and alpha2-adrenergic receptors (alpha2-ARs, Kis = 28, 1. and 1. nM for alpha2A, alpha2B, and alpha2C, respectively). It is selective for these receptors over 5-HT1D (Ki = 2 µM) and 5-HT1B at 10 µM. Spiroxatrine also induces...
| Schlagworte: | R-5188, 8-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one |
| Anwendung: | 5-HT1A/alpha2-AR antagonist |
| CAS | 1054-88-2 |
| MW: | 379.45 D |
ab 118,00 €
Spiroxatrine
Artikelnummer: TGM-T23382-100mg
Description: Spiroxatrine (R 5188) is a selective and potent 5-HT1alpha and alpha2-adrenergic dual antagonist with sedative activity, and inhibitory effects on 5-HT1alpha, 5-HT1beta, 5-HT2, and dopamine receptors. Spiroxatrine may be used in the study of disorders related to the cardiovascular system. Target:...
| Schlagworte: | R 5188 |
| CAS | 1054-88-2 |
| MW: | 379.45 D |
ab 76,00 €
