ENPP1 Inhibitor C

ENPP1 inhibitor C is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1, IC50 = 0.26 µM in a cell-free assay). It is selective for ENPP1 over ENPP2-7 at 10 µM. ENPP1 inhibitor C decreases ENPP1 activity in MDA-MB-231 human breast and C6 rat glioma cancer cells when used at a concentration of 10 µM.Formal Name: 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine. CAS Number: 2378640-92-5. Molecular Formula: C15H18N6. Formula Weight: 282.3. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 30 mg/ml, DMSO: 30 mg/ml, Ethanol: 30 mg/ml. lambdamax: 231 nm. SMILES: NC1=CC=CC(CC2=C(N(C)C)N3C(N=C2C)=NC=N3)=C1. InChi Code: InChI=1S/C15H18N6/c1-10-13(8-11-5-4-6-12(16)7-11)14(20(2)3)21-15(19-10)17-9-18-21/h4-7,9H,8,16H2,1-3H3. InChi Key: VUDSCOCEYOZLJD-UHFFFAOYSA-N.