Fosaprepitant dimeglumine

Fosaprepitant dimeglumine
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay24034-5 5 mg -

6 - 10 business days*

84.00€
Cay24034-10 10 mg -

6 - 10 business days*

129.00€
Cay24034-25 25 mg -

6 - 10 business days*

302.00€
Cay24034-50 50 mg -

6 - 10 business days*

520.00€
 
Fosaprepitant dimeglumine is a water-soluble prodrug form of the neurokinin-1 receptor antagonist... more
Product information "Fosaprepitant dimeglumine"
Fosaprepitant dimeglumine is a water-soluble prodrug form of the neurokinin-1 receptor antagonist aprepitant (Cay-14867). Formulations containing fosaprepitant dimeglumine have been used to prevent chemotherapy-induced nausea and vomiting.Formal Name: 1-deoxy-1-(methylamino)-D-glucitol, [3-[[(2R,3S)-2-[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy]-3-(4-fluorophenyl)-4-morpholinyl]methyl]-2,5-dihydro-5-oxo-1H-1,2,4-triazol-1-yl]phosphonate (2:1). CAS Number: 265121-04-8. Synonyms: MK 0517. Molecular Formula: C23H22F7N4O6P . 2C7H17NO5. Formula Weight: 1004.8. Purity: >95%. Formulation: (Request formulation change), A crystalline solid. Solubility: PBS (pH 7.2): 10 mg/ml. SMILES: FC1=CC=C([C@@H]2N(CC3=NN(P(O)(O)=O)C(N3)=O)CCO[C@@H]2O[C@H](C)C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)C=C1.CNC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO.CNC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO. InChi Code: InChI=1S/C23H22F7N4O6P.2C7H17NO5/c1-12(14-8-15(22(25,26)27)10-16(9-14)23(28,29)30)40-20-19(13-2-4-17(24)5-3-13)33(6-7-39-20)11-18-31-21(35)34(32-18)41(36,37)38,2*1-8-2-4(10)6(12)7(13)5(11)3-9/h2-5,8-10,12,19-20H,6-7,11H2,1H3,(H,31,32,35)(H2,36,37,38),2*4-13H,2-3H2,1H3/t12-,19+,20-,2*4-,5+,6+,7+/m100/s1. InChi Key: VRQHBYGYXDWZDL-OOZCZQCLSA-N.
Keywords: MK 0517, 1-deoxy-1-(methylamino)-D-glucitol, [3-[[(2R,3S)-2-[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy]-3-(4-fluorophenyl)-4-morpholinyl]methyl]-2,5-dihydro-5-oxo-1H-1,2,4-triazol-1-yl]phosphonate (2:1)
Supplier: Cayman Chemical
Supplier-Nr: 24034

Properties

Application: Neurokinin-1 receptor antagonist prodrug
MW: 1004.8 D
Formula: C23H22F7N4O6P . 2C7H17NO5
Purity: >95%
Format: Crystalline Solid

Database Information

CAS : 265121-04-8| Matching products
KEGG ID : K04222 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Signal Word: Danger
GHS Hazard Pictograms:
H Phrases: H302, H315, H318, H373, H400, H410
P Phrases: P260, P264, P270, P273, P280, P301+310, P302+352, P305+351+338, P310, P314, P321, P330, P332+313, P362+364, P391, P501
Caution
Our products are for laboratory research use only: Not for administration to humans!
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